SCHEMBL19334381

SCHEMBL19334381

O=C1NS(=O)(=O)c2cc3c(cc21)C(=O)NS3(=O)=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 16/20 0.59
CA9 Q16790 16/20 0.59
RET P07949 2/20 0.59
GRK5 P34947 2/20 0.59
TYRO3 Q06418 2/20 0.59
DYRK1B Q9Y463 2/20 0.59
CHEK1 O14757 1/20 0.59
DAPK3 O43293 1/20 0.59
MAP4K4 O95819 1/20 0.59
PIM1 P11309 1/20 0.59
LTK P29376 1/20 0.59
CSNK1A1 P48729 1/20 0.59
CDK8 P49336 1/20 0.59
PRKX P51817 1/20 0.59
LIMK1 P53667 1/20 0.59
CDK5 Q00535 1/20 0.59
ACVR1 Q04771 1/20 0.59
PTK2 Q05397 1/20 0.59
PRKAA1 Q13131 1/20 0.59
DYRK1A Q13627 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13931179 0.92 CA12 (0.61) CA12CA9RETGRK5TYRO3
SCHEMBL29587067 0.84 CA12 (0.53) CA12CA9RETGRK5TYRO3
SCHEMBL31503491 0.78 CA12 (0.47) CA12CA9RETGRK5TYRO3
SCHEMBL20529344 0.76 CA12 (0.46) CA12CA9RETGRK5TYRO3
SCHEMBL1249735 0.74 CA12 (0.62) CA12CA9RETGRK5TYRO3
SCHEMBL1290860 0.74 CA12 (1.00) CA12CA9RETGRK5TYRO3
SCHEMBL6753007 0.74 CHEK1 (0.79) CA12CA9RETGRK5TYRO3
SCHEMBL10815413 0.74 CA12 (0.62) CA12CA9RETGRK5TYRO3
SCHEMBL31168119 0.74 CHEK1 (0.79) CA12CA9RETGRK5TYRO3
SCHEMBL29349483 0.74 CA12 (0.62) CA12CA9RETGRK5TYRO3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9757375-B2 Compounds that inhibit human DNA ligases and methods of treating cancer UNIVERSITY OF MARYLAND, BALTIMORE (US) 2017-09-12 US disclosed