SCHEMBL1933716

SCHEMBL1933716

CC(C)c1ccc(-c2n[nH]c(=O)c3ccccc23)cc1.CC(C)c1ccc(-c2nn(N)c(=O)c3ccccc23)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 9/20 0.51
ROCK2 O75116 5/20 0.51
ATM Q13315 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
LMNA P02545 1/20 0.46
TSHR P16473 1/20 0.46
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 1/20 0.46
POLB P06746 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
ALOX15 P16050 1/20 0.46
HSD17B10 Q99714 1/20 0.46
NCOA1 Q15788 1/20 0.45
NCOA3 Q9Y6Q9 1/20 0.45
MAPK1 P28482 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
PDE4A P27815 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1786120 0.90 NPSR1 (0.46) ATMNPSR1LMNAALDH1A1GAA
SCHEMBL1932753 0.86 NPSR1 (0.54) ROCK1ROCK2ATMNPSR1LMNA
SCHEMBL1931814 0.86 ATM (0.54) ROCK1ROCK2ATMNPSR1LMNA
SCHEMBL1788381 0.86 ATM (0.67) ROCK1ROCK2ATMNPSR1LMNA
SCHEMBL1934226 0.83 PDE4A (0.52) ROCK1ROCK2ATMNPSR1LMNA
SCHEMBL24000703 0.78 ATM (0.63) ROCK1ROCK2ATMNPSR1LMNA
SCHEMBL24000505 0.78 ATM (0.63) ROCK1ROCK2ATMNPSR1LMNA
Hydrochloric Acid SCHEMBL30088932 0.77 ATM (0.61) ROCK1ROCK2ATMNPSR1LMNA
Hydrochloric Acid SCHEMBL30088836 0.77 ATM (0.61) ROCK1ROCK2ATMNPSR1LMNA
SCHEMBL8864712 0.75 HPGD (0.63) NPSR1KDM4EALDH1A1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2504317-A1 POTASSIUM CHANNEL MODULATORS Abbott Laboratories (US) 2012-10-03 EP disclosed
WO-2011066168-A1 POTASSIUM CHANNEL MODULATORS ABBOTT LABORATORIES (US) 2011-06-03 WO disclosed