SCHEMBL19337799

SCHEMBL19337799

COc1cc(C(=O)NC(=S)Nc2cccc(NC(=O)C3CCCCCC3)c2)cc(OC)c1OC

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMO Q99835 8/20 0.67
ALDH1A1 P00352 4/20 0.57
MAPT P10636 3/20 0.57
ALOX12 P18054 2/20 0.57
LMNA P02545 2/20 0.57
KDM4E B2RXH2 1/20 0.57
RECQL P46063 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
CYP2C9 P11712 1/20 0.54
TSHR P16473 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.53
GAA P10253 1/20 0.53
KCNK3 O14649 1/20 0.53
KCNK9 Q9NPC2 1/20 0.53
SIRT5 Q9NXA8 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12129851 1.00 SMO (0.67) SMOALDH1A1MAPTALOX12LMNA
SCHEMBL8223133 0.88 TSHR (0.54) SMOALDH1A1LMNATDP1TSHR
SCHEMBL1342152 0.84 MEN1 (0.60) ALDH1A1MAPTALOX12LMNATDP1
SCHEMBL19337794 0.84 TSHR (0.49) SMOALDH1A1LMNATDP1TSHR
SCHEMBL15492188 0.82 KCNK3 (0.49) SMOALDH1A1TSHRKCNK3KCNK9
SCHEMBL19326789 0.81 SMO (0.61) SMOALDH1A1MAPTALOX12LMNA
SCHEMBL1336819 0.81 SMO (0.83) SMOALDH1A1MAPTALOX12LMNA
SCHEMBL29390703 0.81 SMO (1.00) SMOALDH1A1MAPTALOX12LMNA
SCHEMBL12129860 0.81 SMO (1.00) SMOALDH1A1MAPTALOX12LMNA
SCHEMBL19326792 0.80 SMO (0.85) SMOALDH1A1MAPTALOX12LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2291352-B1 N-ACYLTHIOUREA AND N-ACYLUREA INHIBITORS OF THE HEDGEHOG PROTEIN SIGNALLING PATHWAY CENTRE NAT RECH SCIENT (FR) 2017-09-13 EP disclosed