SCHEMBL19339170

SCHEMBL19339170

CC(=O)N1CCCCCC/C=C\c2ccc(NC(=O)c3c[nH]c4ccccc4c3=O)cc21

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CFTR P13569 19/20 0.51
GABRA1 P14867 1/20 0.51
GABRB1 P18505 1/20 0.51
GABRA5 P31644 1/20 0.51
GABRA3 P34903 1/20 0.51
GABRA2 P47869 1/20 0.51
GABRB2 P47870 1/20 0.51
GABRA4 P48169 1/20 0.51
GABRA6 Q16445 1/20 0.51
MAOB P27338 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16327339 0.84 CFTR (0.58) CFTRGABRA1GABRB1GABRA5GABRA3
SCHEMBL22417516 0.84 CFTR (0.58) CFTRGABRA1GABRB1GABRA5GABRA3
SCHEMBL16254149 0.84 CFTR (0.58) CFTRGABRA1GABRB1GABRA5GABRA3
SCHEMBL18708419 0.82 CFTR (0.60) CFTRGABRA1GABRB1GABRA5GABRA3
SCHEMBL396530 0.81 CFTR (0.53) CFTRGABRA1GABRB1GABRA5GABRA3
SCHEMBL394813 0.80 CFTR (0.62) CFTRGABRA1GABRB1GABRA5GABRA3
SCHEMBL2971418 0.75 CFTR (0.69) CFTRGABRA1GABRB1GABRA5GABRA3
SCHEMBL399165 0.74 CFTR (0.55) CFTRGABRA1GABRB1GABRA5GABRA3
SCHEMBL2964947 0.74 CFTR (0.70) CFTRGABRA1GABRB1GABRA5GABRA3
SCHEMBL399479 0.74 CFTR (0.61) CFTRGABRA1GABRB1GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3216787-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2017-09-13 EP disclosed