SCHEMBL19339458

SCHEMBL19339458

CC(C)(C)OC(=O)N1CCC[C@@H]1c1ncc(-c2ccc3cc(Br)ccc3c2)[nH]1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PRCP P42785 8/20 0.49
CYP3A4 P08684 4/20 0.47
CYP2C9 P11712 3/20 0.47
NR1I2 O75469 2/20 0.47
ABCB11 O95342 1/20 0.47
OPRK1 P41145 1/20 0.47
KCNH2 Q12809 1/20 0.47
HPGDS O60760 3/20 0.47
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 1/20 0.44
HCRTR1 O43613 3/20 0.44
HCRTR2 O43614 3/20 0.44
USP30 Q70CQ3 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL204592 1.00 PRCP (0.49) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL2709055 1.00 PRCP (0.49) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL2709400 0.94 PRCP (0.54) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL15511859 0.93 PRCP (0.44) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL2707745 0.92 PRCP (0.52) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL12965885 0.92 PRCP (0.52) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL2757500 0.92 CYP3A4 (0.54) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL203107 0.92 CYP3A4 (0.54) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL2710848 0.92 CYP3A4 (0.54) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL9912059 0.91 PRCP (0.55) PRCPCYP3A4CYP2C9NR1I2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3002281-B1 ANTIVIRAL COMPOUNDS GILEAD PHARMASSET LLC (US) 2017-09-13 EP disclosed