SCHEMBL19339652

SCHEMBL19339652

CC(C)(C)OC(=O)N1CCC[C@H]1c1ncc(-c2ccc3c(c2)oc2cc(-c4ccc5nc(C6CCCN6)[nH]c5c4)ccc23)[nH]1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 2/20 0.42
SCN10A Q9Y5Y9 1/20 0.41
HCRTR1 O43613 13/20 0.40
HCRTR2 O43614 13/20 0.40
PRCP P42785 2/20 0.40
CHEK2 O96017 1/20 0.38
ABCB11 O95342 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
OPRK1 P41145 1/20 0.38
KCNH2 Q12809 1/20 0.38
HPGDS O60760 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2710075 0.94 NR1I2 (0.45) NR1I2HCRTR1HCRTR2PRCPCHEK2
SCHEMBL205289 0.94 NR1I2 (0.45) NR1I2HCRTR1HCRTR2PRCPCHEK2
SCHEMBL12075270 0.91 SCN10A (0.44) NR1I2SCN10AHCRTR1HCRTR2PRCP
SCHEMBL10201491 0.91 SCN10A (0.46) NR1I2SCN10AHCRTR1HCRTR2PRCP
SCHEMBL27978678 0.91 PRCP (0.44) NR1I2HCRTR1HCRTR2PRCPCHEK2
SCHEMBL8749325 0.90 HCRTR1 (0.44) NR1I2SCN10AHCRTR1HCRTR2PRCP
SCHEMBL19339621 0.87 SCN10A (0.52) SCN10AHCRTR1HCRTR2CHEK2
SCHEMBL18462513 0.86 PRCP (0.50) NR1I2HCRTR1HCRTR2PRCPABCB11
SCHEMBL2709583 0.86 PRCP (0.50) NR1I2HCRTR1HCRTR2PRCPABCB11
SCHEMBL204446 0.86 PRCP (0.50) NR1I2HCRTR1HCRTR2PRCPABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3309157-A1 ANTIVIRAL COMPOUNDS Gilead Pharmasset LLC (US) 2018-04-18 EP disclosed
EP-3002281-B1 ANTIVIRAL COMPOUNDS GILEAD PHARMASSET LLC (US) 2017-09-13 EP disclosed