SCHEMBL19339705

SCHEMBL19339705

CC(C)(C)OC(=O)N1CCC[C@H]1c1ncc(-c2ccc3c(c2)S(=O)(=O)c2cc(-c4cnc([C@@H]5CCCN5)[nH]4)ccc2-3)[nH]1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PRCP P42785 11/20 0.46
CYP3A4 P08684 3/20 0.42
CYP2C9 P11712 3/20 0.42
NR1I2 O75469 2/20 0.42
ABCB11 O95342 1/20 0.42
OPRK1 P41145 1/20 0.42
KCNH2 Q12809 1/20 0.42
HPGDS O60760 3/20 0.41
CYP1A2 P05177 2/20 0.40
CYP2D6 P10635 1/20 0.40
HCRTR1 O43613 2/20 0.38
HCRTR2 O43614 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18462732 0.93 PRCP (0.51) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL2708760 0.93 PRCP (0.51) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL20055396 0.89 PRCP (0.45) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL690389 0.88 CYP3A4 (0.52) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL13148034 0.88 CYP3A4 (0.52) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL204049 0.88 CYP3A4 (0.52) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL690388 0.88 CYP3A4 (0.52) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL19339750 0.87 PRCP (0.43) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL203069 0.86 PRCP (0.46) PRCPCYP3A4CYP2C9NR1I2ABCB11
SCHEMBL15368177 0.86 PRCP (0.47) PRCPCYP3A4CYP2C9NR1I2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3309157-A1 ANTIVIRAL COMPOUNDS Gilead Pharmasset LLC (US) 2018-04-18 EP disclosed
EP-3002281-B1 ANTIVIRAL COMPOUNDS GILEAD PHARMASSET LLC (US) 2017-09-13 EP disclosed