SCHEMBL1934759

SCHEMBL1934759

COc1c(NC(=O)c2ccc(Cl)c(Oc3ccnc(CN4CCCN(OC(=O)OC(C)(C)C)CC4)c3)c2)cc(C(C)(C)C)cc1NS(C)(=O)=O

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 17/20 0.44
SRC P12931 9/20 0.42
SYK P43405 8/20 0.42
MAPK14 Q16539 6/20 0.42
BRAF P15056 2/20 0.41
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1936807 0.98 GSK3A (0.44) GSK3ASRCSYKMAPK14BRAF
SCHEMBL1935715 0.93 BRAF (0.45) GSK3ASRCSYKMAPK14BRAF
SCHEMBL1935735 0.91 BRAF (0.47) GSK3ASRCSYKMAPK14BRAF
SCHEMBL1935542 0.91 BRAF (0.43) BRAF
SCHEMBL2671208 0.90 GSK3A (0.45) GSK3ASRCSYKMAPK14BRAF
SCHEMBL1936189 0.90 GSK3A (0.54) GSK3ASRCSYKMAPK14BRAF
SCHEMBL2671149 0.89 GSK3A (0.45) GSK3ASRCSYKMAPK14BRAF
SCHEMBL1936348 0.88 GSK3A (0.52) GSK3ASRCSYKMAPK14BRAF
SCHEMBL1936808 0.88 BRAF (0.49) GSK3ASRCSYKMAPK14BRAF
SCHEMBL1936684 0.88 BRAF (0.45) BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2331506-B1 NOVEL BENZAMIDES, PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM INT (DE) 2013-07-03 EP disclosed
EP-2331506-A1 NOVEL BENZAMIDES, PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS Boehringer Ingelheim International GmbH (DE) 2011-06-15 EP disclosed
WO-2010026095-A1 NOVEL BENZAMIDES, PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-03-11 WO disclosed