SCHEMBL19360702

SCHEMBL19360702

C=CC(=O)Nc1cccc(Oc2nc(Nc3ccc(OC)c(C)c3OC)ncc2Br)c1

nearest known ligand 0.88

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.88
BTK Q06187 1/20 0.63
ITK Q08881 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5585427 0.94 EGFR (1.00) EGFRBTK
SCHEMBL19360705 0.92 EGFR (0.74) EGFRBTKITK
SCHEMBL5585407 0.92 EGFR (1.00) EGFRBTKITK
SCHEMBL19360701 0.90 EGFR (0.88) EGFRBTKITK
SCHEMBL19360700 0.89 EGFR (0.86) EGFRBTKITK
SCHEMBL5585132 0.88 EGFR (1.00) EGFRBTKITK
SCHEMBL19360699 0.87 EGFR (0.87) EGFRITK
SCHEMBL9923761 0.86 EGFR (0.83) EGFRBTKITK
SCHEMBL9923765 0.84 EGFR (0.82) EGFRBTKITK
SCHEMBL5585393 0.84 EGFR (1.00) EGFRBTKITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9765038-B2 Heteroaryl compounds and uses thereof CELGENE CAR LLC (BM) 2017-09-19 US disclosed