SCHEMBL19364299

SCHEMBL19364299

COC(=O)c1cc(Cl)c(C)nn1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 4/20 0.42
MAPK1 P28482 2/20 0.41
NQO2 P16083 4/20 0.40
ALDH1A1 P00352 1/20 0.40
ATM Q13315 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29595828 0.83 NOTUM (0.43) NOTUMMAPK1NQO2ALDH1A1MRGPRX4
SCHEMBL15633295 0.83 NOTUM (0.43) NOTUMMAPK1NQO2ALDH1A1MRGPRX4
SCHEMBL15633243 0.81 NOTUM (0.42) NOTUMMAPK1NQO2ALDH1A1MRGPRX4
SCHEMBL20321125 0.81 MAPK1 (0.43) MAPK1ALDH1A1ATM
SCHEMBL24386910 0.80 NOTUM (0.43) NOTUMMAPK1NQO2ALDH1A1MRGPRX4
SCHEMBL17440068 0.76 NQO2 (0.48) NOTUMMAPK1NQO2ALDH1A1MRGPRX4
SCHEMBL18725396 0.76 NQO2 (0.46) NOTUMMAPK1NQO2ALDH1A1MRGPRX4
SCHEMBL3936135 0.73 MAPK1 (0.47) NOTUMMAPK1NQO2ALDH1A1ATM
SCHEMBL30031450 0.73 MAPK1 (0.47) NOTUMMAPK1NQO2ALDH1A1ATM
SCHEMBL19835436 0.72 MAPK1 (0.50) NOTUMMAPK1NQO2ALDH1A1MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2903977-B1 5-PHENOXY-3H-PYRIMIDIN-4-ONE DERIVATIVES AND THEIR USE AS HIV REVERSE TRANSCRIPTASE INHIBITORS MERCK SHARP & DOHME (US) 2017-09-20 EP disclosed