SCHEMBL19367174

SCHEMBL19367174

COCCONC(=O)c1cc2snnc2c(F)c1Nc1ccc(I)cc1F

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.58
CAMK2B Q13554 1/20 0.58
MAP2K1 Q02750 19/20 0.56
MAP2K2 P36507 1/20 0.55
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
HDAC3 O15379 1/20 0.51
HDAC4 P56524 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC7 Q8WUI4 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC10 Q969S8 1/20 0.51
HDAC11 Q96DB2 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
HDAC9 Q9UKV0 1/20 0.51
HDAC5 Q9UQL6 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15129748 0.92 MAP2K1 (0.67) MAP2K1MAP2K2CYP3A4CYP2C9CYP2C19
SCHEMBL15129746 0.91 MAP2K1 (0.52) PIM1CAMK2BMAP2K1MAP2K2CYP3A4
SCHEMBL16305603 0.86 MEN1 (0.60) PIM1CAMK2BMAP2K1MAP2K2CYP3A4
SCHEMBL19367389 0.86 PIM1 (0.58) PIM1CAMK2BMAP2K1MAP2K2HDAC3
SCHEMBL15129745 0.85 MAP2K1 (0.69) MAP2K1MAP2K2
SCHEMBL15130253 0.85 MAP2K1 (0.48) PIM1CAMK2BMAP2K1MAP2K2CYP3A4
SCHEMBL15131443 0.84 MAP2K1 (0.62) PIM1CAMK2BMAP2K1MAP2K2CYP3A4
SCHEMBL15129550 0.83 MAP2K1 (0.53) PIM1CAMK2BMAP2K1MAP2K2CYP3A4
SCHEMBL19366603 0.83 MAP2K1 (0.53) MAP2K1MAP2K2CYP3A4CYP2C9CYP2C19
SCHEMBL19366620 0.83 MAP2K1 (0.43) PIM1CAMK2BMAP2K1MAP2K2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2804855-B1 BENZOHETEROCYCLIC COMPOUNDS AND USE THEREOF SHANGHAI KECHOW PHARMA INC (CN) 2017-09-20 EP disclosed