SCHEMBL19367408

SCHEMBL19367408

Cc1ccc(Nc2c(C(=O)NOCC(O)CO)cc3scnc3c2F)c(F)c1

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 19/20 0.54
MAP2K2 P36507 4/20 0.54
MAPK1 P28482 2/20 0.54
BRAF P15056 1/20 0.54
MAP2K5 Q13163 1/20 0.54
ABCB11 O95342 1/20 0.45
NQO2 P16083 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15129660 0.90 MAP2K1 (0.69) MAP2K1MAP2K2MAPK1BRAFMAP2K5
SCHEMBL19367194 0.88 MAP2K1 (0.49) MAP2K1MAP2K2MAPK1BRAFMAP2K5
SCHEMBL19366765 0.88 MAP2K1 (0.56) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL19366605 0.86 MAP2K1 (0.54) MAP2K1MAP2K2MAPK1BRAFMAP2K5
SCHEMBL19366614 0.84 MEN1 (0.54) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL15129595 0.83 MAP2K1 (0.56) MAP2K1MAP2K2MAPK1BRAFMAP2K5
SCHEMBL19367201 0.83 MAP2K1 (0.55) MAP2K1MAP2K2MAPK1BRAFMAP2K5
SCHEMBL14590532 0.83 MAP2K1 (0.66) MAP2K1MAP2K2MAPK1BRAFMAP2K5
SCHEMBL19366598 0.82 MAP2K1 (0.44) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL18457665 0.82 MAP2K1 (0.78) MAP2K1MAP2K2MAPK1BRAFMAP2K5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9937158-B2 Benzoheterocyclic compounds and use thereof SHANGHAI KECHOW PHARMA, INC. (CN) 2018-04-10 US disclosed
EP-2804855-B1 BENZOHETEROCYCLIC COMPOUNDS AND USE THEREOF SHANGHAI KECHOW PHARMA INC (CN) 2017-09-20 EP disclosed