SCHEMBL1936896

SCHEMBL1936896

CNC(=O)c1c(-c2ccc(F)cc2)oc2ncc(-c3ccccc3C(=O)O)cc12

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.44
CYP2C8 P10632 4/20 0.44
KCNH2 Q12809 2/20 0.43
NR1I2 O75469 1/20 0.43
ALOX5AP P20292 1/20 0.42
FEN1 P39748 1/20 0.42
BRS3 P32247 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1936301 0.82 TYRO3 (0.46) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL18809708 0.79 CYP3A4 (0.44) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL1935982 0.77 NEK1 (0.46) CYP3A4CYP2C8KCNH2
SCHEMBL1919452 0.76 CYP3A4 (0.55) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL1935460 0.76 CYP3A4 (0.41) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL17464377 0.76 CYP3A4 (0.58) CYP3A4CYP2C8KCNH2
SCHEMBL1935043 0.76 CYP3A4 (0.42) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL17108305 0.75 CYP3A4 (0.49) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL2562440 0.75 CYP2C8 (0.47) CYP3A4CYP2C8KCNH2NR1I2
SCHEMBL17464384 0.75 CYP3A4 (0.46) CYP3A4CYP2C8KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2331502-A2 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2011-06-15 EP disclosed
WO-2010030538-A2 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2010-03-18 WO disclosed