SCHEMBL1937486

SCHEMBL1937486

CCc1cc(-c2c(CC3CC3)nc3ccc(N4CCN[C@H](C)C4)nn23)ccn1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CSNK1E P49674 6/20 0.54
PIM1 P11309 3/20 0.37
ZAP70 P43403 3/20 0.36
PRKD1 Q15139 2/20 0.36
PRKD2 Q9BZL6 2/20 0.36
PIM3 Q86V86 1/20 0.36
PIM2 Q9P1W9 1/20 0.36
PRKCQ Q04759 1/20 0.35
PRKCD Q05655 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1937484 1.00 CSNK1E (0.54) CSNK1EPIM1ZAP70PRKD1PRKD2
SCHEMBL477091 0.90 CSNK1E (0.54) CSNK1EPIM1ZAP70PRKD1PRKD2
SCHEMBL477092 0.90 CSNK1E (0.54) CSNK1EPIM1ZAP70PRKD1PRKD2
SCHEMBL477176 0.87 CSNK1E (0.69) CSNK1E
SCHEMBL477143 0.87 CSNK1E (0.69) CSNK1E
SCHEMBL477023 0.83 CSNK1E (0.59) CSNK1EPIM1
SCHEMBL477025 0.83 CSNK1E (0.59) CSNK1EPIM1
SCHEMBL477061 0.80 CSNK1E (0.73) CSNK1E
SCHEMBL477060 0.80 CSNK1E (0.73) CSNK1E
SCHEMBL477034 0.77 CSNK1E (0.59) CSNK1EPIM1ZAP70PRKD1PRKD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2331546-A1 2-ALKYL-6-CYCLOAMINO-3-(PYRIDIN-4-YL)IMIDAZO[1,2-IB]-PYRIDAZINE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC APPLICATION THEREOF Sanofi-aventis (FR) 2011-06-15 EP claimed
WO-2010018327-A1 2-ALKYL-6-CYCLOAMINO-3-(PYRIDIN-4-YL)IMIDAZO[1,2-IB]-PYRIDAZINE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC APPLICATION THEREOF SANOFI-AVENTIS (FR) 2010-02-18 WO claimed