SCHEMBL1937680

SCHEMBL1937680

COCC(C)Nc1nc(Nc2ccc(S(=O)(=O)N(C)C)cc2)ncc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 13/20 0.48
CDK1 P06493 12/20 0.48
CDK2 P24941 12/20 0.48
SYK P43405 2/20 0.47
CDK4 P11802 3/20 0.46
CA2 P00918 2/20 0.46
CDK7 P50613 2/20 0.46
CDK9 P50750 2/20 0.46
CCNT1 O60563 1/20 0.46
CCND1 P24385 1/20 0.46
CCNH P51946 1/20 0.46
CCNB1 P14635 1/20 0.46
CCNE1 P24864 1/20 0.46
AXL P30530 3/20 0.44
AURKA O14965 1/20 0.44
AURKB Q96GD4 1/20 0.44
NEK2 P51955 1/20 0.44
EGFR P00533 1/20 0.42
STK17B O94768 1/20 0.41
STK17A Q9UEE5 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4065488 0.88 CDK1 (0.62) KDRCDK1CDK2CDK4CA2
Hydrochloric Acid SCHEMBL2444643 0.80 AURKA (0.44) KDRCDK1CDK2CDK4CA2
SCHEMBL4063041 0.76 CDK1 (0.77) KDRCDK1CDK2CDK4CA2
SCHEMBL4062176 0.75 CDK1 (0.63) KDRCDK1CDK2CDK4CA2
SCHEMBL1937120 0.74 JAK3 (0.47) SYKEGFR
SCHEMBL1916775 0.74 STK17A (0.51) SYKSTK17BSTK17A
SCHEMBL29832995 0.71 PTK2 (0.59) CDK7CDK9AXLAURKAAURKB
SCHEMBL4065206 0.71 CDK1 (0.62) KDRCDK1CDK2CDK4CA2
SCHEMBL1474421 0.71 BCL6 (0.63) KDRSYKAURKAAURKBEGFR
SCHEMBL1935476 0.70 KDM4E (0.45) CDK2SYKSTK17BSTK17A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2330904-A2 4-ALKYL-SUBSTITUTED DIAMINOPYRIMIDINES Bayer CropScience AG (DE) 2011-06-15 EP disclosed
WO-2010025863-A2 4-ALKYL-SUBSTITUTED DIAMINOPYRIMIDINES BAYER CROPSCIENCE AG (DE) 2010-03-11 WO disclosed