SCHEMBL1938155

SCHEMBL1938155

NC(=O)O[C@@H](Cc1ccccc1)[C@@H](O)CNCc1cccc(C(F)(F)F)c1

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 17/20 0.60
BCHE P06276 4/20 0.60
CTSD P07339 13/20 0.51
BACE2 Q9Y5Z0 12/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1938153 1.00 BACE1 (0.60) BACE1BCHECTSDBACE2
SCHEMBL3343893 0.86 BACE1 (0.56) BACE1BCHECTSDBACE2
SCHEMBL8580373 0.85 BCHE (0.52) BACE1BCHE
SCHEMBL3343882 0.81 BACE1 (0.55) BACE1BCHECTSDBACE2
SCHEMBL8276492 0.81 BACE1 (0.62) BACE1BCHECTSDBACE2
SCHEMBL161260 0.81 BACE1 (0.62) BACE1BCHECTSDBACE2
SCHEMBL3455222 0.81 BACE1 (0.62) BACE1BCHECTSDBACE2
SCHEMBL1937520 0.80 BACE1 (0.47) BACE1CTSD
SCHEMBL1937521 0.80 BACE1 (0.47) BACE1CTSD
Hydrochloric Acid SCHEMBL2499284 0.80 BACE1 (0.61) BACE1BCHECTSDBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2185561-B1 1,2,3,4-tetrahydropyrrolo(1,2-a)pyrazine-6-carboxamide and 2,3,4,5-tetrahydropyrrolo(1,2-a)-diazepine-7-carboxamide derivatives, preparation and therapeutic use thereof SANOFI AVENTIS (FR) 2011-06-15 EP disclosed