SCHEMBL19406491

SCHEMBL19406491

O=C(O)N1CCN(C(=O)Cn2cc(Nc3ncc(Cl)c(NCc4ccccc4)n3)cn2)CC1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 14/20 0.65
JAK2 O60674 7/20 0.53
JAK1 P23458 6/20 0.53
TTK P33981 3/20 0.53
TYK2 P29597 2/20 0.53
KDR P35968 1/20 0.51
AURKB Q96GD4 1/20 0.51
AURKA O14965 1/20 0.51
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC10 Q969S8 1/20 0.50
HDAC11 Q96DB2 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
HDAC9 Q9UKV0 1/20 0.50
HDAC5 Q9UQL6 1/20 0.50
NTRK1 P04629 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16812321 0.94 JAK3 (0.66) JAK3JAK2JAK1TTKTYK2
SCHEMBL19417616 0.93 JAK3 (0.63) JAK3JAK2JAK1TTKTYK2
SCHEMBL15546244 0.91 JAK3 (0.63) JAK3JAK2JAK1TTKTYK2
SCHEMBL16782469 0.91 JAK3 (0.77) JAK3JAK2JAK1TTKTYK2
SCHEMBL19406496 0.91 JAK3 (0.58) JAK3JAK2JAK1TTKTYK2
SCHEMBL15547137 0.89 JAK3 (0.59) JAK3JAK2JAK1TTKTYK2
SCHEMBL15547232 0.88 JAK3 (0.63) JAK3JAK2JAK1TTKTYK2
SCHEMBL15548500 0.88 JAK3 (0.57) JAK3JAK2JAK1TTKTYK2
SCHEMBL15547437 0.87 JAK3 (0.64) JAK3JAK2JAK1TTKTYK2
SCHEMBL15546726 0.86 JAK3 (0.62) JAK3JAK2JAK1TTKTYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2855451-B1 HETEROCYCLYL PYRIMIDINE ANALOGUES AS TYK2 INHIBITORS CELLZOME LTD (GB) 2017-10-04 EP claimed