SCHEMBL19418317

SCHEMBL19418317

O=C1/C=C/CCC(O)CC[C@H](c2ccccc2)OC(=O)c2c(O)cc(O)c(Cl)c2C1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 4/20 0.56
MAPT P10636 3/20 0.43
HSP90AA1 P07900 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
HPGD P15428 2/20 0.43
GAA P10253 1/20 0.43
RAB9A P51151 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
NLRP3 Q96P20 1/20 0.43
CBR1 P16152 1/20 0.43
PTGS2 P35354 1/20 0.43
ACLY P53396 1/20 0.43
FTO Q9C0B1 1/20 0.43
ALDH1A1 P00352 1/20 0.43
F13A1 P00488 1/20 0.39
TGM2 P21980 1/20 0.39
CYP1A1 P04798 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP19A1 P11511 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10150867 0.85 HSP90AB1 (0.58) HSP90AB1MAPTHSP90AA1MEN1KMT2A
SCHEMBL10150018 0.85 HSP90AB1 (0.70) HSP90AB1MAPTHSP90AA1MEN1KMT2A
SCHEMBL10150021 0.85 HSP90AB1 (0.70) HSP90AB1MAPTHSP90AA1MEN1KMT2A
SCHEMBL10150124 0.85 HSP90AB1 (0.73) HSP90AB1MAPTHSP90AA1MEN1KMT2A
SCHEMBL19418321 0.82 HSP90AB1 (0.61) HSP90AB1MAPTHSP90AA1MEN1KMT2A
SCHEMBL14293412 0.82 HSP90AB1 (0.58) HSP90AB1MAPTHSP90AA1MEN1KMT2A
SCHEMBL19418251 0.75 HSP90AB1 (0.57) HSP90AB1MAPTHSP90AA1MEN1KMT2A
SCHEMBL10150081 0.75 HSP90AB1 (0.76) HSP90AB1MAPTHSP90AA1MEN1KMT2A
SCHEMBL14155841 0.74 HSP90AB1 (0.72) HSP90AB1MAPTHSP90AA1MEN1KMT2A
SCHEMBL10150859 0.74 HSP90AB1 (0.75) HSP90AB1MAPTHSP90AA1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2136799-B1 MACROCYCLIC COMPOUNDS USEFUL AS INHIBITORS OF KINASES AND HSP90 UNIV STRASBOURG (FR) 2017-10-04 EP disclosed