SCHEMBL19418385

SCHEMBL19418385

O=C1/C=C/CC2CC(C[C@H](c3ccccc3)OC(=O)c3c(O)cc(O)cc3C1)O2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F13A1 P00488 1/20 0.49
TGM2 P21980 1/20 0.49
CYP19A1 P11511 3/20 0.42
CYP3A4 P08684 3/20 0.42
CYP1A1 P04798 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP1B1 Q16678 2/20 0.42
MEN1 O00255 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
KMT2A Q03164 2/20 0.42
HSD17B10 Q99714 2/20 0.42
MAPT P10636 2/20 0.42
CYP2D6 P10635 1/20 0.42
MKNK2 Q9HBH9 3/20 0.37
MKNK1 Q9BUB5 1/20 0.37
HSP90AB1 P08238 3/20 0.37
KIT P10721 4/20 0.36
PDGFRA P16234 4/20 0.36
KDR P35968 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19417979 1.00 F13A1 (0.49) F13A1TGM2CYP19A1CYP3A4CYP1A1
SCHEMBL19418153 0.83 F13A1 (0.64) F13A1TGM2CYP3A4MAPTMKNK2
SCHEMBL10150026 0.82 F13A1 (0.57) F13A1TGM2CYP19A1CYP3A4CYP1A1
SCHEMBL19418453 0.82 F13A1 (0.57) F13A1TGM2CYP19A1CYP3A4CYP1A1
SCHEMBL10150031 0.82 F13A1 (0.57) F13A1TGM2CYP19A1CYP3A4CYP1A1
SCHEMBL10150126 0.82 F13A1 (0.55) F13A1TGM2CYP19A1CYP3A4CYP1A1
SCHEMBL10150131 0.82 F13A1 (0.55) F13A1TGM2CYP19A1CYP3A4CYP1A1
SCHEMBL10150865 0.81 F13A1 (0.56) F13A1TGM2CYP19A1CYP3A4CYP1A1
SCHEMBL10150870 0.81 F13A1 (0.56) F13A1TGM2CYP19A1CYP3A4CYP1A1
SCHEMBL19418053 0.73 F13A1 (0.44) F13A1TGM2CYP19A1CYP3A4CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2136799-B1 MACROCYCLIC COMPOUNDS USEFUL AS INHIBITORS OF KINASES AND HSP90 UNIV STRASBOURG (FR) 2017-10-04 EP disclosed