SCHEMBL19447155

SCHEMBL19447155

Cc1cncc(C(C)Nc2cccc(C(C)Nc3cncc(Cl)n3)c2)c1

nearest known ligand 0.69

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 15/20 0.69
RET P07949 1/20 0.63
PDGFRB P09619 1/20 0.63
KIT P10721 1/20 0.63
SRC P12931 1/20 0.63
PDGFRA P16234 1/20 0.63
FLT1 P17948 1/20 0.63
FLT4 P35916 1/20 0.63
KDR P35968 1/20 0.63
FRK P42685 1/20 0.63
DDR1 Q08345 1/20 0.63
CDK2 P24941 1/20 0.41
LDHA P00338 1/20 0.39
LDHB P07195 1/20 0.39
KDM4E B2RXH2 1/20 0.39
PFKFB3 Q16875 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13340049 1.00 CSF1R (0.69) CSF1RRETPDGFRBKITSRC
SCHEMBL3478309 0.93 CSF1R (0.72) CSF1RRETPDGFRBKITSRC
SCHEMBL19447154 0.84 CSF1R (0.67) CSF1RRETPDGFRBKITSRC
SCHEMBL19447153 0.84 CSF1R (0.67) CSF1RRETPDGFRBKITSRC
SCHEMBL3474393 0.83 CSF1R (0.77) CSF1RRETPDGFRBKITSRC
SCHEMBL3474546 0.82 CSF1R (1.00) CSF1RRETPDGFRBKITSRC
SCHEMBL29119452 0.82 CSF1R (1.00) CSF1RRETPDGFRBKITSRC
SCHEMBL30672146 0.82 CSF1R (1.00) CSF1RRETPDGFRBKITSRC
SCHEMBL13340116 0.78 CSF1R (1.00) CSF1RRETPDGFRBKITSRC
SCHEMBL13340142 0.78 CSF1R (0.87) CSF1RRETPDGFRBKITSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2848610-B1 Inhibitors of kinase activity YM BIOSCIENCES AUSTRALIA PTY (AU) 2017-10-11 EP disclosed