SCHEMBL19447232

SCHEMBL19447232

CC(Nc1cncc(-c2ccc(CN3CCN(C)CC3)cc2)n1)c1cccc(NC(=O)c2cccc(C(F)(F)F)c2)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 13/20 0.65
BRAF P15056 2/20 0.55
FGFR1 P11362 1/20 0.51
DDR2 Q16832 1/20 0.51
SRC P12931 3/20 0.49
PDGFRB P09619 2/20 0.49
PDGFRA P16234 2/20 0.49
RET P07949 1/20 0.49
KIT P10721 1/20 0.49
FLT1 P17948 1/20 0.49
FLT4 P35916 1/20 0.49
KDR P35968 1/20 0.49
FRK P42685 1/20 0.49
DDR1 Q08345 1/20 0.49
JAK2 O60674 1/20 0.47
ABL1 P00519 1/20 0.46
BCR P11274 1/20 0.46
SYK P43405 1/20 0.46
BTK Q06187 1/20 0.45
ACKR3 P25106 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13340409 1.00 CSF1R (0.65) CSF1RBRAFFGFR1DDR2SRC
SCHEMBL3475477 0.92 CSF1R (0.64) CSF1RBRAFSRCPDGFRBPDGFRA
SCHEMBL3475478 0.92 CSF1R (0.64) CSF1RBRAFSRCPDGFRBPDGFRA
SCHEMBL13340272 0.89 CSF1R (0.65) CSF1RBRAFFGFR1DDR2SRC
SCHEMBL3475141 0.87 CSF1R (0.71) CSF1RSRCPDGFRBPDGFRARET
SCHEMBL3475138 0.87 CSF1R (0.71) CSF1RSRCPDGFRBPDGFRARET
SCHEMBL13340286 0.86 CSF1R (0.63) CSF1RBRAFSRCPDGFRBPDGFRA
SCHEMBL13340431 0.86 CSF1R (0.61) CSF1RBRAFSRCPDGFRBPDGFRA
SCHEMBL18023931 0.85 ABL1 (0.64) CSF1RBRAFDDR2SRCPDGFRB
SCHEMBL17954640 0.84 CSF1R (0.73) CSF1RSRCPDGFRBPDGFRARET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2848610-B1 Inhibitors of kinase activity YM BIOSCIENCES AUSTRALIA PTY (AU) 2017-10-11 EP disclosed