SCHEMBL19447262

SCHEMBL19447262

COc1cccc(-c2cncc(NC(C)c3cccc(NC(=O)c4cccc(C)c4)c3)n2)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 15/20 0.71
RET P07949 1/20 0.71
PDGFRB P09619 1/20 0.71
KIT P10721 1/20 0.71
SRC P12931 1/20 0.71
PDGFRA P16234 1/20 0.71
FLT1 P17948 1/20 0.71
FLT4 P35916 1/20 0.71
KDR P35968 1/20 0.71
FRK P42685 1/20 0.71
DDR1 Q08345 1/20 0.71
LDHA P00338 1/20 0.56
LDHB P07195 1/20 0.56
KCNK3 O14649 1/20 0.55
KCNK9 Q9NPC2 1/20 0.55
PFKFB3 Q16875 1/20 0.52
BRAF P15056 1/20 0.52
MEN1 O00255 1/20 0.50
MAPT P10636 1/20 0.50
KMT2A Q03164 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13340136 1.00 CSF1R (0.71) CSF1RRETPDGFRBKITSRC
SCHEMBL13339898 0.93 CSF1R (0.71) CSF1RRETPDGFRBKITSRC
SCHEMBL20101067 0.90 CSF1R (0.72) CSF1RRETPDGFRBKITSRC
SCHEMBL19447209 0.90 CSF1R (0.57) CSF1RRETPDGFRBKITSRC
SCHEMBL13340157 0.90 CSF1R (0.57) CSF1RRETPDGFRBKITSRC
SCHEMBL13339859 0.90 CSF1R (0.79) CSF1RRETPDGFRBKITSRC
SCHEMBL13340082 0.88 CSF1R (0.82) CSF1RRETPDGFRBKITSRC
SCHEMBL13339927 0.88 CSF1R (0.72) CSF1RRETPDGFRBKITSRC
SCHEMBL19447211 0.88 CSF1R (0.72) CSF1RRETPDGFRBKITSRC
SCHEMBL20101087 0.87 CSF1R (0.70) CSF1RRETPDGFRBKITSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2848610-B1 Inhibitors of kinase activity YM BIOSCIENCES AUSTRALIA PTY (AU) 2017-10-11 EP disclosed