SCHEMBL19456591

SCHEMBL19456591

N=C(N)N/N=C1\c2cc(OC(F)(F)F)ccc2-n2c1nc1ncccc1c2=O

nearest known ligand 0.66

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 18/20 0.66
CXCR3 P49682 2/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20597235 1.00 IDO1 (0.66) IDO1CXCR3CYP3A4
SCHEMBL20597091 0.91 IDO1 (0.66) IDO1
SCHEMBL19456598 0.91 IDO1 (0.66) IDO1
SCHEMBL24777808 0.87 IDO1 (0.72) IDO1CXCR3CYP3A4
SCHEMBL20597269 0.84 IDO1 (0.62) IDO1
SCHEMBL30141703 0.84 IDO1 (0.62) IDO1
SCHEMBL19456484 0.84 IDO1 (0.62) IDO1
SCHEMBL20597579 0.81 IDO1 (0.67) IDO1
SCHEMBL19456434 0.81 IDO1 (0.67) IDO1
SCHEMBL30141744 0.81 IDO1 (0.67) IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017173973-A1 NITROGEN HETEROCYCLIC TRYPTAMINE KETONE DERIVATIVE AND APPLICATION AS IDO1 AND/OR TDO INHIBITOR 北京大学 2017-10-12 WO disclosed