SCHEMBL194645

SCHEMBL194645

NC(O)CCc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 2/20 0.57
ERAP1 Q9NZ08 2/20 0.57
ERAP2 Q6P179 1/20 0.57
METAP2 P50579 1/20 0.49
METAP1 P53582 1/20 0.49
CYP2A6 P11509 1/20 0.48
HTR2A P28223 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
TAAR1 Q96RJ0 1/20 0.48
LOXL2 Q9Y4K0 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
EPHX1 P07099 1/20 0.46
ACP3 P15309 1/20 0.46
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
SLC6A3 Q01959 2/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1760865 1.00 ANPEP (0.57) ANPEPERAP1ERAP2METAP2METAP1
SCHEMBL4282969 1.00 ANPEP (0.57) ANPEPERAP1ERAP2METAP2METAP1
Hydrochloric Acid SCHEMBL28675057 0.98 ANPEP (0.55) ANPEPERAP1ERAP2METAP2METAP1
Hydrochloric Acid SCHEMBL20590185 0.98 ANPEP (0.55) ANPEPERAP1ERAP2METAP2METAP1
Hydrochloric Acid SCHEMBL16988 0.98 ANPEP (0.55) ANPEPERAP1ERAP2METAP2METAP1
Sulfuric Acid SCHEMBL1605647 0.90 BLM (0.55) ANPEPERAP1ERAP2METAP2METAP1
Nitric Acid SCHEMBL7055225 0.87 ANPEP (0.50) ANPEPERAP1ERAP2METAP2METAP1
SCHEMBL7998233 0.86 GRIK1 (0.54) ANPEPERAP1ERAP2HTR2ASMN1; SMN2
SCHEMBL456442 0.86 GRIK1 (0.54) ANPEPERAP1ERAP2HTR2ASMN1; SMN2
SCHEMBL14544283 0.86 GRIK1 (0.54) ANPEPERAP1ERAP2HTR2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2075 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3607938-B1 PHARMACEUTICAL COMPOSITION SOVIC BRKICIC LJILJANA (HR) 2026-05-27 EP claimed
EP-4209246-B1 METHOD OF MANUFACTURING OF A PARTICLE-ATTACHED MICRONEEDLE QUADMEDICINE INC (KR) 2026-02-18 EP claimed
EP-3968065-B1 PLANAR LIGHTING DEVICE LG ELECTRONICS INC (KR) 2025-05-28 EP claimed
EP-1773302-B2 RAPIDLY DISINTEGRATING GELATINOUS COATED TABLETS JOHNSON & JOHNSON CONSUMER INC (US) 2024-06-26 EP claimed
EP-4380942-A1 NOVEL APPLICATIONS FOR OXAZABOROLIDINES AND NEW METHODS OF MANUFACTURE THEREOF Pathway Intermediates Limited (GB) 2024-06-12 EP claimed
CN-113880721-B Synthesis method of dapoxetine 湖南九典制药股份有限公司 2024-05-28 CN claimed
CN-117736399-A Bio-based polyurethane foam based on lignin oligomer and vegetable oil and preparation method thereof 中国林业科学研究院林产化学工业研究所 2024-03-22 CN claimed
US-20230392750-A1 HIGH-PRESSURE COMPOSITE CONTAINER YAPP AUTOMOTIVE SYSTEMS CO., LTD (CN) 2023-12-07 US claimed
EP-3697386-B1 LIQUID COMPOSITIONS FOR PERORAL USE COMPRISING PHOSPHATIDYLGLYCEROL DERIVATIVES AND THIXOTROPIC EXCIPIENTS FOR TREATING CARDIAC CHANNELOPATHIES CAUSED BY PHARMACOLOGICAL AGENTS SIGNPATH PHARMA INC (US) 2023-07-26 EP claimed
EP-4206516-A1 HIGH-PRESSURE COMPOSITE CONTAINER Yapp Automotive Systems Co., Ltd. (CN) 2023-07-05 EP claimed
EP-0132472-B1 MEDICATED PRODUCTS CONTAINING A MAGNESIUM TRISILICATE ADSORBENT WITH A MEDICAMENT DRUG ADSORBED THEREON WARNER-LAMBERT COMPANY (US) 1989-06-21 EP claimed
EP-0139881-B1 LIQUID PROLONGED RELEASE PHARMACEUTICAL FORMULATIONS CONTAINING IONIC CONSTITUENTS PENNWALT CORPORATION (US) 1989-05-10 EP claimed
EP-0123585-B1 TRANSDERMAL DRUG FORM RHONE-POULENC SANTE (FR) 1988-08-31 EP claimed
EP-0097523-B1 EXTENDED ACTION CONTROLLED RELEASE COMPOSITIONS Euroceltique S.A. (LU) 1988-01-13 EP claimed
US-4639368-A CARBON DIOXIDE GENERATOR FARMACON RESEARCH CORPORATION (US) 1987-01-27 US claimed
EP-0173928-A1 Controlled-release medical preparations AB LEO (SE) 1986-03-12 EP claimed
EP-0152379-A2 Process for preparing pharmaceutical compositions containing unilamellar liposomes CIBA-GEIGY AG (CH) 1985-08-21 EP claimed
US-4522984-A WITH E-CAPROLACTONE DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1985-06-11 US claimed
EP-0036145-B1 AN ORALLY ADMINISTERED DRUG FORM COMPRISING A POLAR BIOACTIVE AGENT AND AN ADJUVANT INTERx RESEARCH CORPORATION (US) 1985-05-29 EP claimed
US-4045450-A Optical resolution of DL-pantolactone ALPS PHARMACEUTICAL IND. CO., LTD. (JA) 1977-08-30 US claimed