SCHEMBL19485461

SCHEMBL19485461

Cc1cc(N(C)CCN(C)C)c([N+](=O)[O-])cc1Nc1ncc(C(=O)OC(C)C)c(-c2cn(C)c3ncccc23)n1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.57
ERBB2 P04626 1/20 0.54
ERBB3 P21860 1/20 0.54
ERBB4 Q15303 1/20 0.54
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19103353 0.92 EGFR (0.67) EGFRERBB2ERBB3ERBB4
SCHEMBL19103343 0.92 EGFR (0.64) EGFRERBB2ERBB3ERBB4KCNH2
SCHEMBL19320679 0.92 EGFR (0.53) EGFRERBB2ERBB3ERBB4
SCHEMBL19320677 0.89 EGFR (0.59) EGFRERBB2ERBB3ERBB4KCNH2
SCHEMBL19103315 0.88 EGFR (0.47) EGFRERBB2ERBB3ERBB4KCNH2
SCHEMBL19103323 0.86 EGFR (0.65) EGFRERBB2ERBB3ERBB4KCNH2
SCHEMBL19103256 0.86 EGFR (0.65) EGFRERBB2ERBB3ERBB4KCNH2
SCHEMBL19103272 0.86 EGFR (0.51) EGFRERBB2ERBB3ERBB4
SCHEMBL17384966 0.86 EGFR (0.62) EGFRERBB2ERBB3ERBB4KCNH2
SCHEMBL19103351 0.86 EGFR (0.57) EGFRERBB2ERBB3ERBB4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9796712-B2 Heteroaryl compounds for kinase inhibition ARIAD PHARMACEUTICALS, INC. (US) 2017-10-24 US disclosed