SCHEMBL19485463

SCHEMBL19485463

CCn1cc(-c2nc(Nc3cc([N+](=O)[O-])c(F)cc3C)ncc2C(=O)OC)c2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGFR P00533 16/20 0.48
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
NR4A2 P43354 1/20 0.41
MKNK2 Q9HBH9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19103274 0.93 EGFR (0.53) EGFR
SCHEMBL19493392 0.92 EGFR (0.57) EGFRMKNK2
SCHEMBL19103273 0.89 EGFR (0.61) EGFR
SCHEMBL19103275 0.87 EGFR (0.48) EGFRMKNK2
SCHEMBL19485460 0.87 EGFR (0.58) EGFR
SCHEMBL19103265 0.87 EGFR (0.58) EGFR
SCHEMBL19103269 0.83 EGFR (0.57) EGFR
SCHEMBL19103271 0.83 EGFR (0.44) EGFR
SCHEMBL19103293 0.82 EGFR (0.51) EGFR
SCHEMBL30748688 0.82 EGFR (0.63) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9796712-B2 Heteroaryl compounds for kinase inhibition ARIAD PHARMACEUTICALS, INC. (US) 2017-10-24 US disclosed