SCHEMBL19489684

SCHEMBL19489684

Cc1cccc(F)c1Oc1nc(NC2CCCC2)cc(-c2ccc(=O)n(C)c2)n1

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 8/20 0.44
CREBBP Q92793 10/20 0.42
MAP3K12 Q12852 1/20 0.36
EGLN1 Q9GZT9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19489676 0.90 BRD4 (0.54) BRD4CREBBPMAP3K12
SCHEMBL19489527 0.85 CREBBP (0.52) BRD4CREBBP
SCHEMBL19460471 0.85 PFKFB3 (0.51) BRD4
SCHEMBL19489535 0.85 PFKFB3 (0.51) BRD4
SCHEMBL19490107 0.85 PFKFB3 (0.51) BRD4
SCHEMBL19489832 0.84 PFKFB3 (0.45) BRD4CREBBP
SCHEMBL19489833 0.84 CREBBP (0.53) BRD4CREBBP
SCHEMBL19489824 0.82 CREBBP (0.51) BRD4CREBBP
SCHEMBL19489782 0.82 CREBBP (0.49) BRD4CREBBP
SCHEMBL19490108 0.82 CREBBP (0.52) BRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10202360-B2 Therapeutic compounds CELGENE QUANTICEL RESEARCH, INC. (US) 2019-02-12 US disclosed
US-20170298040-A1 THERAPEUTIC COMPOUNDS CELGENE QUANTICEL RESEARCH, INC. 2017-10-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10202360-B2 Therapeutic compounds EP300, BRDT, BRPF3 BRD4 5/4885CREBBP 32/4885MAP3K12 487/4885
US-20170298040-A1 THERAPEUTIC COMPOUNDS EP300, BRDT, BRPF3 BRD4 5/4885CREBBP 32/4885MAP3K12 487/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.