SCHEMBL19554378

SCHEMBL19554378

COC(=O)c1cc(Cl)c(C#C[Si](C)(C)C)cc1N

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.48
ALDH1A1 P00352 6/20 0.48
GAA P10253 4/20 0.48
ABL1 P00519 1/20 0.47
HSD17B10 Q99714 3/20 0.41
HPGD P15428 3/20 0.41
MAPT P10636 2/20 0.41
GLA P06280 2/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
ATM Q13315 1/20 0.41
NQO2 P16083 6/20 0.40
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
CFTR P13569 5/20 0.39
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21857652 0.88 GAA (0.42) KDM4EALDH1A1GAAABL1HSD17B10
SCHEMBL2012660 0.84 CA12 (0.41) KDM4EGAAABL1NQO2TSHR
SCHEMBL23015343 0.83 KDM4E (0.51) KDM4EALDH1A1GAAABL1HSD17B10
SCHEMBL149267 0.83 GAA (0.44) KDM4EALDH1A1GAAABL1HSD17B10
SCHEMBL29511129 0.80 KDM4E (0.45) KDM4EALDH1A1GAAABL1HSD17B10
SCHEMBL2391826 0.77 CFTR (0.58) KDM4EALDH1A1GAAABL1HSD17B10
SCHEMBL1884944 0.77 GAA (0.64) KDM4EALDH1A1GAAABL1HSD17B10
SCHEMBL30344983 0.76 KDM4E (0.42) KDM4EALDH1A1GAAABL1HSD17B10
SCHEMBL28183743 0.76 ABL1 (0.38) KDM4EALDH1A1GAAABL1HPGD
SCHEMBL25156545 0.76 KDM4E (0.42) KDM4EALDH1A1GAAABL1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed