SCHEMBL19602

SCHEMBL19602

CC(=O)Nc1cc[c]cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.60
L3MBTL1 Q9Y468 2/20 0.60
HTT P42858 1/20 0.60
NAPRT Q6XQN6 1/20 0.60
HSD17B10 Q99714 1/20 0.60
KMT2A Q03164 6/20 0.58
MEN1 O00255 3/20 0.58
ALDH1A1 P00352 3/20 0.58
MAPT P10636 2/20 0.58
CA12 O43570 2/20 0.58
CA1 P00915 2/20 0.58
CA2 P00918 2/20 0.58
CA9 Q16790 2/20 0.58
TDP1 Q9NUW8 1/20 0.58
BRD4 O60885 1/20 0.58
NR1I2 O75469 1/20 0.58
MB P02144 1/20 0.58
CYP1A1 P04798 1/20 0.58
CA3 P07451 1/20 0.58
CYP3A4 P08684 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28349149 0.98 SMN1; SMN2 (0.58) SMN1; SMN2L3MBTL1HTTNAPRTHSD17B10
SCHEMBL27742196 0.98 SMN1; SMN2 (0.58) SMN1; SMN2L3MBTL1HTTNAPRTHSD17B10
SCHEMBL3140177 0.87 SMN1; SMN2 (0.76) SMN1; SMN2L3MBTL1HTTNAPRTHSD17B10
SCHEMBL10883881 0.87 CACNA1B (0.69) SMN1; SMN2L3MBTL1HTTKMT2AMEN1
SCHEMBL4490164 0.83 KMT2A (0.46) SMN1; SMN2L3MBTL1HTTNAPRTHSD17B10
SCHEMBL1283740 0.82 KMT2A (0.59) SMN1; SMN2L3MBTL1HTTKMT2AMEN1
SCHEMBL861674 0.82 SMN1; SMN2 (0.84) SMN1; SMN2L3MBTL1HTTNAPRTHSD17B10
SCHEMBL5037216 0.81 KDM1A (0.69) SMN1; SMN2L3MBTL1KMT2AMEN1ALDH1A1
SCHEMBL342425 0.79 RXFP1 (0.58) SMN1; SMN2L3MBTL1HTTNAPRTHSD17B10
SCHEMBL3398708 0.78 KDM1A (0.67) SMN1; SMN2L3MBTL1KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 8886 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118344284-A Compound with benzamide structure and preparation method and application thereof 杭州医学院 2024-07-16 CN claimed
WO-2024146922-A1 C5AR1 INHIBITORS FOR USE IN THE TREATMENT OF OCULAR MUCOUS MEMBRANE PEMPHIGOID AND/OR ORAL MUCOUS MEMBRANE PEMPHIGOID DOMPE' FARMACEUTICI SPA (IT) 2024-07-11 WO claimed
EP-4397306-A1 C5AR1 INHIBITORS FOR USE IN THE TREATMENT OF OCULAR MUCOUS MEMBRANE PEMPHIGOID AND/OR ORAL MUCOUS MEMBRANE PEMPHIGOID Dompe' Farmaceutici S.P.A. (IT) 2024-07-10 EP claimed
US-20240217913-A2 PREPARATION OF SUBSTITUTED ACRYLATE COMPOUND HUA MEDICINE (SHANGHAI) LTD. (CN) 2024-07-04 US claimed
CN-118221577-A 2-Phenoxyquinoline derivative, and preparation method and application thereof 湖南中医药大学 2024-06-21 CN claimed
US-20240180888-A1 C5AR1 INHIBITORS FOR TREATING HYPERSENSITIVITY REACTIONS TO TAXANES DOMPE' FARMACEUTICI SPA (IT) 2024-06-06 US claimed
US-11987588-B2 Modulators of the beta-3 adrenergic receptor useful for the treatment or prevention of heart failure and disorders related thereto ARENA PHARMACEUTICALS, INC. (US) 2024-05-21 US claimed
EP-4357344-A2 SUBSTITUTED PYRIDAZINONES AS HERBICIDES Syngenta Crop Protection AG (CH) 2024-04-24 EP claimed
US-20240116903-A1 TETRAHYDROQUINOLINE DERIVATIVE AND MEDICINAL USE THEREOF TORAY INDUSTRIES, INC. (JP) 2024-04-11 US claimed
CN-117843543-A Preparation method of alpha, alpha-difluorobutyrolactam 南京工业大学 2024-04-09 CN claimed
US-4011208-A 3-CYANO OR ACYL-4-ARYL-5-ARYLAZO-6-HYDROXYPYRIDONE-2 DYES SANDOZ LTD. (CH) 1977-03-08 US claimed
US-3998803-A TEXTILES FIDELITY UNION TRUST COMPANY, EXECUTIVE TRUSTEE UNDER THE SANDOZ TRUST (US) 1976-12-21 US claimed
US-3978223-A UREIDOACETAMIDO-PENICILLINS FOR TREATING BACTERIAL INFECTIONS BAYER AKTIENGESELLSCHAFT (DT) 1976-08-31 US claimed
US-3971784-A ANTIMETABOLITES MITSUI PHARMACEUTICALS, INCORPORATED (JA) 1976-07-27 US claimed
US-3966703-A Asymmetrical frisazo dyestuffs derived from diazotized 2,7-diamino-carbazole BAYER AKTIENGESELLSCHAFT (DT) 1976-06-29 US claimed
US-3950327-A NEW NITRONES, THEIR MANUFACTURE AND THEIR USE FOR THE MANUFACTURE OF N-SUBSTITUTED ARALIPHATIC ALDEHYDE-NITRONES CIBA-GEIGY CORPORATION (US) 1976-04-13 US claimed
US-3948939-A 9-Acyl-1,2,3,4-tetrahydrocarbazole-3 and 4-carboxylic acids STERLING DRUG INC. (US) 1976-04-06 US claimed
US-3947516-A Novel aromatic aldehydes and process for preparing them HOECHST AKTIENGESELLSCHAFT (DT) 1976-03-30 US claimed
US-3943120-A WATER INSOLUBLE CIBA-GEIGY AG (CH) 1976-03-09 US claimed
US-3933795-A Ureidoacetamido-penicillins Konig, Hans-Bodo (DT) 1976-01-20 US claimed