SCHEMBL19610508

SCHEMBL19610508

NC(=O)c1ccc(Oc2ccc3c(c2)COB3O)cc1.O=C(O)C1CCCC1

nearest known ligand 0.66

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 15/20 0.66
PDE4A P27815 12/20 0.66
PDE4C Q08493 12/20 0.66
PDE4D Q08499 12/20 0.66
CHRM1 P11229 1/20 0.51
ADRA1A P35348 1/20 0.51
PDE1A P54750 1/20 0.51
PDE3B Q13370 1/20 0.51
PDE7A Q13946 1/20 0.51
PDE3A Q14432 1/20 0.51
KLK1 P06870 1/20 0.49
KLK5 Q9Y337 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2529448 0.89 PDE4B (0.78) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL5583359 0.80 PDE4B (1.00) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL595819 0.80 PDE4B (1.00) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL2530321 0.78 PDE4B (0.65) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL11993084 0.77 PDE4B (0.78) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL2530713 0.76 PDE4B (0.73) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL2531912 0.76 PDE4B (0.56) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL2529550 0.76 PDE4B (0.68) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL2526209 0.75 PDE4B (0.55) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL30571023 0.75 PDE4B (1.00) PDE4BPDE4APDE4CPDE4DCHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246034-A1 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2017-11-22 EP disclosed