SCHEMBL19617010

SCHEMBL19617010

COC[C@@H]1CN(c2nc(OC[C@@H]3CCCN3C)nc3c2CCNC3)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KRAS P01116 20/20 0.45
VHL P40337 1/20 0.41
CDK7 P50613 1/20 0.41
CCNH P51946 1/20 0.41
MNAT1 P51948 1/20 0.41
SOS1 Q07889 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19637617 1.00 KRAS (0.45) KRASVHLCDK7CCNHMNAT1
SCHEMBL19948569 1.00 KRAS (0.45) KRASVHLCDK7CCNHMNAT1
SCHEMBL19959367 0.95 KRAS (0.45) KRASVHLCDK7CCNHMNAT1
SCHEMBL30188633 0.95 KRAS (0.45) KRASVHLCDK7CCNHMNAT1
SCHEMBL29246035 0.95 KRAS (0.45) KRASVHLCDK7CCNHMNAT1
SCHEMBL19964238 0.91 KRAS (0.44) KRASVHLCDK7CCNHMNAT1
SCHEMBL19616467 0.91 KRAS (0.56) KRASVHLCDK7CCNHMNAT1
SCHEMBL19617279 0.91 KRAS (0.56) KRASVHLCDK7CCNHMNAT1
SCHEMBL30188819 0.91 KRAS (0.56) KRASVHLCDK7CCNHMNAT1
SCHEMBL19616721 0.91 KRAS (0.56) KRASVHLCDK7CCNHMNAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3710439-A1 KRAS G12C INHIBITORS Mirati Therapeutics, Inc. (US) 2020-09-23 EP disclosed
EP-3458445-A1 KRAS G12C INHIBITORS Mirati Therapeutics, Inc. (US) 2019-03-27 EP disclosed
WO-2017201161-A1 KRAS G12C INHIBITORS Mirati Therapeutics, Inc. (US) 2017-11-23 WO disclosed