SCHEMBL19620645

SCHEMBL19620645

NC1=C(OS(=O)Cc2ccccc2)C(=O)C(c2ccc(F)c(F)c2)O1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
GRM5 P41594 1/20 0.32
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19620558 0.90 KDM4E (0.34) KDM4EPOLBMAPT
SCHEMBL15627599 0.87 KDM4E (0.41) KDM4EPOLBMAPT
SCHEMBL22902083 0.87 KDM4E (0.39) KDM4EPOLBMAPTGRM5
SCHEMBL19620541 0.86 KDM4E (0.37) KDM4EPOLBMAPTCYP1A2CYP3A4
SCHEMBL19620621 0.86 MAPT (0.49) KDM4EPOLBMAPTCYP1A2CYP3A4
SCHEMBL20367974 0.85 MAPT (0.41) KDM4EPOLBMAPT
SCHEMBL20368252 0.84 MAPT (0.39) KDM4EPOLBMAPTGRM5
SCHEMBL19620595 0.84 KCNA5 (0.36) KDM4EPOLBMAPTCYP1A2CYP3A4
SCHEMBL19620538 0.84 KDM4E (0.37) KDM4EPOLBMAPTCYP1A2CYP3A4
SCHEMBL19620597 0.83 DPP4 (0.38) KDM4EPOLBMAPTGRM5CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2897607-B1 INHIBITORS OF BETA-HYDROLASE FOR TREATMENT OF CANCER RHODE ISLAND HOSPITAL (US) 2017-11-22 EP disclosed