SCHEMBL19620683

SCHEMBL19620683

NC1=C(OS(=O)Cc2ccccc2)C(=O)C(c2cccc(F)c2F)O1

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
KDM1A O60341 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
GRM5 P41594 1/20 0.31
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19620539 0.92 CYP1A2 (0.33) HTR2CHTR2BCYP1A2CYP3A4CYP2C19
SCHEMBL22902013 0.86 CYP1A2 (0.33) HTR2CHTR2BCYP1A2CYP3A4CYP2C19
SCHEMBL19620599 0.85 SMN1; SMN2 (0.33) KDM1APOLB
SCHEMBL19620597 0.83 DPP4 (0.38) CYP1A2CYP3A4CYP2C19GRM5KDM4E
SCHEMBL19620692 0.83 DPP4 (0.38) HTR2CHTR2BCYP1A2CYP3A4CYP2C19
SCHEMBL20368268 0.82 HTR2C (0.34) HTR2CHTR2BCYP1A2CYP3A4CYP2C19
SCHEMBL22902028 0.82 HTR2A (0.34) HTR2CHTR2BCYP1A2CYP3A4CYP2C19
SCHEMBL19620621 0.81 MAPT (0.49) HTR2BCYP1A2CYP3A4CYP2C19KDM4E
SCHEMBL15627599 0.81 KDM4E (0.41) KDM1AKDM4EPOLBMAPT
SCHEMBL22902083 0.80 KDM4E (0.39) KDM1AMAOAMAOBGRM5KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2897607-B1 INHIBITORS OF BETA-HYDROLASE FOR TREATMENT OF CANCER RHODE ISLAND HOSPITAL (US) 2017-11-22 EP disclosed