SCHEMBL19622277

SCHEMBL19622277

CCOC(=O)c1ccc(O)c(Oc2ccc3c(c2)COB3O)c1

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 17/20 0.67
PDE4A P27815 11/20 0.57
PDE4C Q08493 11/20 0.57
PDE4D Q08499 11/20 0.57
HSD17B2 P37059 1/20 0.50
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45
CA9 Q16790 1/20 0.45
CA14 Q9ULX7 1/20 0.45
CHRM1 P11229 1/20 0.45
ADRA1A P35348 1/20 0.45
PDE1A P54750 1/20 0.45
PDE3B Q13370 1/20 0.45
PDE7A Q13946 1/20 0.45
PDE3A Q14432 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2528454 0.92 PDE4B (0.67) PDE4BPDE4APDE4CPDE4DCA12
SCHEMBL2529695 0.89 PDE4B (0.66) PDE4BPDE4APDE4CPDE4DHSD17B2
SCHEMBL2526576 0.87 PDE4B (0.75) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL2526890 0.87 PDE4B (0.66) PDE4BPDE4APDE4CPDE4D
SCHEMBL16478634 0.85 PDE4B (0.64) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL2528794 0.84 PDE4B (0.63) PDE4BPDE4APDE4CPDE4DPDE1A
SCHEMBL8378720 0.84 PDE4B (0.68) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL2527604 0.84 PDE4B (0.60) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL11993006 0.81 PDE4B (0.54) PDE4BPDE4APDE4CPDE4DHSD17B2
SCHEMBL8378196 0.81 PDE4B (0.66) PDE4BPDE4APDE4CPDE4DCHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246034-A1 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2017-11-22 EP disclosed