SCHEMBL19623562

SCHEMBL19623562

O=Nc1cccc(-c2nc(N3CCOCC3)nc3c2CCN3C(=O)Cc2ccccc2)c1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 20/20 0.51
PIK3R1 P27986 5/20 0.49
PIK3CD O00329 1/20 0.42
CYP3A4 P08684 1/20 0.42
AKT1 P31749 1/20 0.42
PIK3CB P42338 1/20 0.42
PIK3CG P48736 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2376517 0.89 PIK3CA (0.66) PIK3CAPIK3R1
SCHEMBL25269771 0.86 PIK3CA (0.58) PIK3CAPIK3R1PIK3CDCYP3A4AKT1
SCHEMBL2378238 0.81 PIK3CA (0.58) PIK3CAPIK3R1AKT1
SCHEMBL2376510 0.80 PIK3CA (0.64) PIK3CAPIK3R1
SCHEMBL19623564 0.80 PIK3CA (0.47) PIK3CAPIK3R1
SCHEMBL19623541 0.78 PIK3CA (0.55) PIK3CAPIK3R1PIK3CBPIK3CG
SCHEMBL2376771 0.77 PIK3CA (0.60) PIK3CAPIK3R1
SCHEMBL2376941 0.77 PIK3CA (0.64) PIK3CAPIK3R1
SCHEMBL3224544 0.76 PIK3CA (0.71) PIK3CAPIK3R1
SCHEMBL12246793 0.75 PIK3CA (0.62) PIK3CAPIK3R1PIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed