SCHEMBL19627741

SCHEMBL19627741

COc1ccc(CN(c2ncns2)S(=O)(=O)c2c(F)cc(F)c(Cl)c2F)c(C)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.38
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
PSEN1 P49768 2/20 0.31
PSEN2 P49810 2/20 0.31
APH1B Q8WW43 2/20 0.31
NCSTN Q92542 2/20 0.31
APH1A Q96BI3 2/20 0.31
PSENEN Q9NZ42 2/20 0.31
SCN1A P35498 1/20 0.31
SCN5A Q14524 1/20 0.31
SCN8A Q9UQD0 1/20 0.31
USP2 O75604 1/20 0.31
TP53 P04637 1/20 0.31
POLB P06746 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19613979 0.91 SCN9A (0.41) SCN9AHDAC8HDAC6SCN1ASCN5A
SCHEMBL19627736 0.89 SCN9A (0.36) SCN9A
SCHEMBL19627659 0.86 SCN1A (0.34) SCN9AHDAC8HDAC6PSEN1PSEN2
SCHEMBL18352341 0.85 SCN9A (0.36) SCN9APSEN1PSEN2APH1BNCSTN
SCHEMBL9923645 0.84 SCN9A (0.38) SCN9A
SCHEMBL19631846 0.83 SCN9A (0.38) SCN9ASCN1ASCN5ASCN8ATP53
SCHEMBL19627592 0.83 SCN9A (0.43) SCN9APSEN1PSEN2APH1BNCSTN
SCHEMBL22088599 0.83 SCN9A (0.41) SCN9AHDAC8TP53POLBGAA
SCHEMBL19631588 0.82 SCN9A (0.37) SCN9AHDAC8SCN1ASCN5ASCN8A
SCHEMBL19613425 0.80 SCN9A (0.39) SCN9AHDAC8USP2TP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170334902-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2017-11-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170334902-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS SCN1A, SCN1B, SCN2B SCN9A 52/4885HDAC8 772/4885HDAC6 537/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.