SCHEMBL19630085

SCHEMBL19630085

Cc1c(C=O)c(=O)n(C2CCCC2)c2nc(Nc3ccc(N4CCNCC4)cn3)ncc12

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.79
CCND1 P24385 18/20 0.79
CCND2 P30279 14/20 0.79
CCND3 P30281 14/20 0.79
CDK2 P24941 5/20 0.76
CCNA2 P20248 4/20 0.76
CDK6 Q00534 4/20 0.76
CCNA1 P78396 3/20 0.76
CDK1 P06493 2/20 0.76
CCNB1 P14635 2/20 0.76
FLT3 P36888 2/20 0.76
CHEK1 O14757 1/20 0.76
DAPK3 O43293 1/20 0.76
CCNT1 O60563 1/20 0.76
CCNT2 O60583 1/20 0.76
ROCK2 O75116 1/20 0.76
STK16 O75716 1/20 0.76
CCNK O75909 1/20 0.76
PDE5A O76074 1/20 0.76
PRKD3 O94806 1/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28412630 0.93 CDK4 (0.78) CDK4CCND1CCND2CCND3CDK2
SCHEMBL4826672 0.88 CDK4 (1.00) CDK4CCND1CCND2CCND3CDK2
SCHEMBL29507539 0.88 CDK4 (1.00) CDK4CCND1CCND2CCND3CDK2
SCHEMBL29507507 0.88 CDK4 (1.00) CDK4CCND1CCND2CCND3CDK2
SCHEMBL6221577 0.88 CDK4 (1.00) CDK4CCND1CCND2CCND3CDK2
SCHEMBL28409617 0.88 CDK4 (0.76) CDK4CCND1CCND2CCND3CDK2
SCHEMBL6223801 0.88 CDK4 (0.98) CDK4CCND1CCND2CCND3CDK2
SCHEMBL15874775 0.87 CDK4 (0.89) CDK4CCND1CCND2CCND3CDK2
SCHEMBL15874369 0.87 CDK4 (0.74) CDK4CCND1CCND2CCND3CDK2
SCHEMBL4828618 0.86 CDK4 (0.80) CDK4CCND1CCND2CCND3CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4289844-A2 A PROCESS FOR MAKING PALBOCICLIB Synthon B.V. (NL) 2023-12-13 EP disclosed
EP-3458604-B1 METHOD FOR DETERMINING SENSITIVITY TO A CDK4/6 INHIBITOR UNIV BRUXELLES (BE) 2021-04-14 EP disclosed
WO-2017198685-A1 METHOD FOR DETERMINING SENSITIVITY TO A CDK4/6 INHIBITOR Université Libre de Bruxelles (BE) 2017-11-23 WO disclosed