SCHEMBL19631574

SCHEMBL19631574

CC(C)CCN(C)[C@@H]1CCN(C2(C(=O)c3ccccn3)CCOC(C)(C)C2)C1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
GRM4 Q14833 3/20 0.34
SMYD3 Q9H7B4 1/20 0.33
TSHR P16473 2/20 0.33
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
MCHR1 Q99705 1/20 0.32
LMNA P02545 3/20 0.31
OPRK1 P41145 1/20 0.31
CTSK P43235 1/20 0.31
CCR5 P51681 2/20 0.31
ICMT O60725 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31
KDM4E B2RXH2 1/20 0.31
CACNA1B Q00975 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19631789 1.00 CYP2D6 (0.35) CYP2D6CYP2C19GRM4SMYD3TSHR
SCHEMBL21221686 1.00 CYP2D6 (0.35) CYP2D6CYP2C19GRM4SMYD3TSHR
SCHEMBL21221659 1.00 CYP2D6 (0.35) CYP2D6CYP2C19GRM4SMYD3TSHR
SCHEMBL21221729 1.00 CYP2D6 (0.35) CYP2D6CYP2C19GRM4SMYD3TSHR
SCHEMBL21221658 1.00 CYP2D6 (0.35) CYP2D6CYP2C19GRM4SMYD3TSHR
SCHEMBL21221660 0.90 GRM4 (0.35) GRM4HPGDMCHR1LMNAALDH1A1
SCHEMBL21221650 0.90 GRM4 (0.35) GRM4HPGDMCHR1LMNAALDH1A1
SCHEMBL21221653 0.90 GRM4 (0.35) GRM4HPGDMCHR1LMNAALDH1A1
SCHEMBL21221667 0.90 GRM4 (0.35) GRM4HPGDMCHR1LMNAALDH1A1
SCHEMBL19631842 0.90 GRM4 (0.35) GRM4HPGDMCHR1LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198339-A1 TETRAHYDROPYRAN AND THIOPYRAN DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2017-11-23 WO disclosed