SCHEMBL19632056

SCHEMBL19632056

CCOCCCN1CCC([C@@]2(C(=O)c3ccccn3)CCOC(C)(C)C2)CC1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 4/20 0.38
HRH2 P25021 1/20 0.38
GRM4 Q14833 3/20 0.36
HRH3 Q9Y5N1 3/20 0.36
OPRM1 P35372 2/20 0.36
HTR1A P08908 2/20 0.35
HTR2A P28223 2/20 0.35
DRD2 P14416 2/20 0.35
DRD3 P35462 2/20 0.35
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19632058 1.00 HRH1 (0.38) HRH1HRH2GRM4HRH3OPRM1
SCHEMBL19632057 0.97 HRH1 (0.39) HRH1HRH2GRM4OPRM1GAA
SCHEMBL19631691 0.90 GRM4 (0.37) HRH1HRH2GRM4HRH3OPRM1
SCHEMBL19631612 0.89 GRM4 (0.37) GRM4OPRM1HTR1AHTR2ADRD2
SCHEMBL19631589 0.88 GRM4 (0.36) HRH1HRH2GRM4HRH3OPRM1
SCHEMBL19631998 0.86 GRM4 (0.38) GRM4OPRM1DRD2
SCHEMBL19631852 0.86 GRM4 (0.38) GRM4OPRM1DRD2
SCHEMBL19631839 0.86 GRM4 (0.38) GRM4OPRM1DRD2
SCHEMBL19631856 0.85 GRM4 (0.36) GRM4
SCHEMBL19631922 0.85 GRM4 (0.36) GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198339-A1 TETRAHYDROPYRAN AND THIOPYRAN DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2017-11-23 WO disclosed