SCHEMBL1963339

SCHEMBL1963339

CCCCn1c(Sc2nc3cc(OC)ccc3s2)nc2c([N])ncnc21

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 18/20 0.62
HSP90AB1 P08238 18/20 0.62
ERBB2 P04626 1/20 0.53
HSP90B1 P14625 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4900283 0.89 HSP90AA1 (0.77) HSP90AA1HSP90AB1ERBB2HSP90B1
SCHEMBL4897565 0.76 HSP90AA1 (1.00) HSP90AA1HSP90AB1HSP90B1
SCHEMBL1964689 0.74 HSP90AA1 (1.00) HSP90AA1HSP90AB1
Ammonia Solution, Strong SCHEMBL6352818 0.72 HSP90AA1 (0.73) HSP90AA1HSP90AB1HSP90B1
SCHEMBL5043365 0.71 HSP90AA1 (1.00) HSP90AA1HSP90AB1HSP90B1
SCHEMBL14466464 0.71 HSP90AA1 (0.82) HSP90AA1HSP90AB1
SCHEMBL3114041 0.71 HSP90AA1 (0.56) HSP90AA1HSP90AB1
SCHEMBL5514963 0.70 HSP90AA1 (1.00) HSP90AA1HSP90AB1
SCHEMBL1964277 0.70 HSP90AA1 (1.00) HSP90AA1HSP90AB1ERBB2HSP90B1
SCHEMBL6897052 0.69 PPARA (0.62)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2336133-A1 Purine analogs having HSP90-inhibiting activity Conforma Therapeutics Corporation (US) 2011-06-22 EP disclosed