SCHEMBL19635078

SCHEMBL19635078

COCc1nn(C)c2c1-c1cccc3c(CCCOc4cccc5ccccc45)c(C=O)n(c13)CCCCCOC2

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 16/20 0.56
BAD Q92934 5/20 0.55
BCL2L1 Q07817 4/20 0.55
BCL2 P10415 3/20 0.49
PMAIP1 Q13794 2/20 0.44
ALB P02768 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19635422 0.90 MCL1 (0.56) MCL1BADBCL2L1BCL2PMAIP1
SCHEMBL19615204 0.89 MCL1 (0.72) MCL1BADBCL2L1BCL2PMAIP1
SCHEMBL19635061 0.88 MCL1 (0.72) MCL1BADBCL2L1BCL2PMAIP1
SCHEMBL24378161 0.87 MCL1 (0.70) MCL1BADBCL2L1BCL2PMAIP1
SCHEMBL19635906 0.87 MCL1 (0.64) MCL1BADBCL2L1BCL2PMAIP1
SCHEMBL19635347 0.86 MCL1 (0.50) MCL1BADBCL2L1BCL2
SCHEMBL19635592 0.86 MCL1 (0.69) MCL1BADBCL2L1BCL2
SCHEMBL19635631 0.86 MCL1 (0.65) MCL1BADBCL2L1BCL2PMAIP1
Diethylamine SCHEMBL19615089 0.86 MCL1 (0.70) MCL1BADBCL2L1BCL2PMAIP1
SCHEMBL24378134 0.84 BAD (0.67) MCL1BADBCL2L1BCL2PMAIP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3458459-B1 MACROCYCLIC INDOLE DERIVATIVES BAYER AG (DE) 2022-04-27 EP disclosed
WO-2017198341-A1 MACROCYCLIC INDOLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2017-11-23 WO disclosed