SCHEMBL19635792

SCHEMBL19635792

Nc1ncnc2c1c(-c1ccc(Oc3ccc(F)cc3F)cc1)nn2[C@@H]1CCCN(C(=O)/C=C/CO)C1

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BTK Q06187 18/20 0.74
EGFR P00533 11/20 0.74
SRC P12931 4/20 0.74
BLK P51451 1/20 0.64
LCK P06239 1/20 0.63
JAK3 P52333 1/20 0.63
ITK Q08881 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28374849 1.00 BTK (0.74) BTKEGFRSRCBLKLCK
SCHEMBL19635198 0.86 BTK (0.55) BTKEGFRSRCBLKLCK
SCHEMBL19635649 0.86 BTK (0.74) BTKEGFRSRCBLKLCK
SCHEMBL19635651 0.86 BTK (0.74) BTKEGFRSRCBLKLCK
SCHEMBL17915683 0.86 EGFR (0.84) BTKEGFRSRCBLKLCK
SCHEMBL18123577 0.85 BTK (0.76) BTKEGFRSRCBLKJAK3
SCHEMBL17173970 0.85 BTK (1.00) BTKEGFRSRC
SCHEMBL17157116 0.85 BTK (1.00) BTKEGFRSRC
SCHEMBL15691524 0.85 BTK (1.00) BTKEGFRSRC
SCHEMBL18700203 0.84 BTK (0.83) BTKEGFRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198049-A1 PYRAZOLOPYRIMIDINE DERIVATIVE AS BTK INHIBITOR AND PREPARATION METHOD AND PHARMACEUTICAL COMPOSITION THEREOF 浙江予川医药科技有限公司 2017-11-23 WO disclosed