SCHEMBL19639035

SCHEMBL19639035

CCOc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1NC(=O)/C=C/CN(C)C

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.66
ERBB2 P04626 8/20 0.66
KDR P35968 8/20 0.64
JAK3 P52333 1/20 0.59
ERBB4 Q15303 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19100193 0.90 EGFR (0.68) EGFRERBB2KDR
Maleic Acid SCHEMBL20637511 0.87 EGFR (0.65) EGFRERBB2KDRERBB4
SCHEMBL19639014 0.86 EGFR (0.87) EGFRERBB2JAK3ERBB4
SCHEMBL30101593 0.86 EGFR (0.87) EGFRERBB2JAK3ERBB4
SCHEMBL5648037 0.85 EGFR (0.69) EGFRERBB2KDRJAK3ERBB4
SCHEMBL5648049 0.85 EGFR (0.69) EGFRERBB2KDRJAK3ERBB4
SCHEMBL26930728 0.84 EGFR (0.78) EGFRERBB2KDRJAK3ERBB4
SCHEMBL2131031 0.82 EGFR (0.87) EGFRERBB2KDRJAK3ERBB4
SCHEMBL2131022 0.82 EGFR (0.87) EGFRERBB2KDRJAK3ERBB4
SCHEMBL19124461 0.81 EGFR (0.63) EGFRERBB2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9957237-B2 Crystal form of neptinib di-p-methylbenzenesulfonate, preparation method thereof, and pharmaceutical composition containing same SHENZHEN NEPTUNUS PHARMACEUTICAL RESEARCH INSTITUTE CO., LTD. (CN) 2018-05-01 US disclosed
US-20170342037-A1 A CRYSTAL FORM OF NEPTINIB di-P-METHYLBENZENESULFONATE, PREPARATION METHOD THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME SHENZHEN NEPTUNUS PHARMACEUTICAL RESEARCH INSTITUTE CO., LTD. (CN) 2017-11-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170342037-A1 A CRYSTAL FORM OF NEPTINIB di-P-METHYLBENZENESULFONATE, PREPARATION METHOD THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME ABL1, NEK5, CYP2D6 EGFR 252/4885ERBB2 874/4885KDR 52/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.