SCHEMBL1964467

SCHEMBL1964467

COc1ccc(I)c(Sc2nc3c(N)nc(F)nc3n2CCC=C(C)C)c1

nearest known ligand 0.77

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 11/20 0.77
HSP90AA1 P07900 11/20 0.53
HSP90AB1 P08238 8/20 0.53
CDC37 Q16543 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1964460 0.90 ERBB2 (0.62) ERBB2HSP90AA1HSP90AB1
SCHEMBL1963481 0.90 ERBB2 (0.78) ERBB2HSP90AA1HSP90AB1CDC37
SCHEMBL1964875 0.87 ERBB2 (1.00) ERBB2HSP90AA1HSP90AB1CDC37
SCHEMBL1963368 0.83 ERBB2 (1.00) ERBB2HSP90AA1HSP90AB1CDC37
SCHEMBL1963254 0.82 HSP90AA1 (0.59) ERBB2HSP90AA1HSP90AB1
SCHEMBL1965154 0.81 ERBB2 (0.64) ERBB2HSP90AA1HSP90AB1
SCHEMBL1966387 0.77 ERBB2 (0.82) ERBB2HSP90AA1HSP90AB1
SCHEMBL1963778 0.76 HSP90AB1 (0.73) ERBB2HSP90AA1HSP90AB1
SCHEMBL5039827 0.74 ERBB2 (0.78) ERBB2HSP90AA1HSP90AB1CDC37
SCHEMBL5038267 0.74 ERBB2 (0.83) ERBB2HSP90AA1HSP90AB1CDC37

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4397691-B2 2010-01-13 JP claimed
JP-2005511565-A 2005-04-28 JP claimed
EP-1440072-A4 PURINE ANALOGS HAVING HSP90-INHIBITING ACTIVITY CONFORMA THERAPEUTIC CORP (US) 2005-02-02 EP claimed
EP-1440072-A2 PURINE ANALOGS HAVING HSP90-INHIBITING ACTIVITY Conforma Therapeutic Corporation (US) 2004-07-28 EP claimed
WO-2003037860-A2 PURINE ANALOGS HAVING HSP90-INHIBITING ACTIVITY CONFORMA THERAPEUTICS CORPORATION (US) 2003-05-08 WO claimed
EP-2336133-A1 Purine analogs having HSP90-inhibiting activity Conforma Therapeutics Corporation (US) 2011-06-22 EP disclosed