SCHEMBL19661007

SCHEMBL19661007

Cc1nc(I)c2sccc2n1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 10/20 0.46
ADORA1 P30542 9/20 0.46
SMN1; SMN2 Q16637 3/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
HTT P42858 1/20 0.38
AXL P30530 1/20 0.37
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
HRH3 Q9Y5N1 1/20 0.36
POLB P06746 1/20 0.36
ALDH1A1 P00352 1/20 0.36
ADORA3 P0DMS8 1/20 0.35
ADORA2B P29275 1/20 0.35
ELANE P08246 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL61008 0.79 ADORA2A (0.49) ADORA2AADORA1SMN1; SMN2RAB9ANPC1
SCHEMBL20458005 0.79 AXL (0.39) ADORA2AADORA1SMN1; SMN2RAB9AHTT
SCHEMBL1367259 0.78 AXL (0.52) ADORA2AADORA1SMN1; SMN2RAB9ANPC1
SCHEMBL24170311 0.76 ADORA2A (0.50) ADORA2AADORA1SMN1; SMN2RAB9ANPC1
SCHEMBL5334843 0.76 ADORA2A (0.50) ADORA2AADORA1SMN1; SMN2RAB9ANPC1
SCHEMBL30277827 0.76 ADORA2A (0.50) ADORA2AADORA1SMN1; SMN2RAB9ANPC1
SCHEMBL24139592 0.76 ADORA2A (0.47) ADORA2AADORA1SMN1; SMN2RAB9ANPC1
Hydrochloric Acid SCHEMBL30277817 0.74 ADORA2A (0.49) ADORA2AADORA1SMN1; SMN2RAB9ANPC1
SCHEMBL10268901 0.73 HTT (0.63) ADORA2AADORA1SMN1; SMN2RAB9ANPC1
SCHEMBL179279 0.73 ADORA2A (0.44) ADORA2AADORA1SMN1; SMN2RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3889152-A1 HETEROAROMATIC DERIVATIVES FOR USE AS REGULATOR, PREPARATION METHOD THEREFOR AND USE THEREOF Jiangsu Hansoh Pharmaceutical Group Co., Ltd. (CN) 2021-10-06 EP disclosed
WO-2017205762-A1 INHIBITORS OF INTERLEUKIN-1 RECEPTOR-ASSOCIATED KINASE PHARMACYCLICS LLC (US) 2017-11-30 WO disclosed