SCHEMBL1966283

SCHEMBL1966283

O=C(O)N1CCC(F)C(Oc2cccc3ccc(-c4nnc5ccccn45)nc23)CC1

nearest known ligand 0.78

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 20/20 0.78
PIM2 Q9P1W9 20/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1968401 0.90 PIM1 (0.74) PIM1PIM2
SCHEMBL1967440 0.89 PIM1 (0.75) PIM1PIM2
SCHEMBL1968348 0.89 PIM2 (0.73) PIM1PIM2
SCHEMBL1977328 0.88 PIM2 (0.84) PIM1PIM2
SCHEMBL1967528 0.88 PIM1 (1.00) PIM1PIM2
SCHEMBL1967531 0.88 PIM1 (1.00) PIM1PIM2
SCHEMBL1967533 0.88 PIM1 (1.00) PIM1PIM2
SCHEMBL1986852 0.86 PIM2 (0.67) PIM1PIM2
SCHEMBL1966057 0.85 PIM2 (0.64) PIM1PIM2
SCHEMBL1967492 0.85 PIM2 (0.64) PIM1PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334677-B1 TRIAZOLOPYRIDINE COMPOUNDS AS PIM KINASE INHIBITORS ARRAY BIOPHARMA INC (US) 2013-10-09 EP disclosed
EP-2334677-A1 TRIAZOLOPYRIDINE COMPOUNDS AS PIM KINASE INHIBITORS Array Biopharma, Inc. (US) 2011-06-22 EP disclosed
WO-2010022076-A1 TRIAZOLOPYRIDINE COMPOUNDS AS PIM KINASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2010-02-25 WO disclosed