SCHEMBL19668445

SCHEMBL19668445

Cc1cccc(C)c1OC[C@H](C)NCCc1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.67
SIGMAR1 Q99720 2/20 0.55
SCN4A P35499 4/20 0.52
SCN8A Q9UQD0 3/20 0.49
LMNA P02545 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
TSHR P16473 1/20 0.49
NFKB1 P19838 1/20 0.49
KCNK3 O14649 1/20 0.49
CACNA1F O60840 1/20 0.49
KCNK2 O95069 1/20 0.49
GBA1 P04062 1/20 0.49
MAOA P21397 1/20 0.49
HTR2A P28223 1/20 0.49
SLC6A4 P31645 1/20 0.49
SCN1A P35498 1/20 0.49
HTR2B P41595 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19668444 1.00 KCNH2 (0.67) KCNH2SIGMAR1SCN4ASCN8ALMNA
SCHEMBL19686658 0.85 SCN4A (0.55) KCNH2SIGMAR1SCN4ASCN8ALMNA
SCHEMBL19668683 0.81 KCNH2 (0.58) KCNH2SIGMAR1SCN4ASCN8ALMNA
SCHEMBL8819029 0.81 KCNH2 (0.58) KCNH2SIGMAR1SCN4ASCN8ALMNA
SCHEMBL7699543 0.81 KCNH2 (0.58) KCNH2LMNANR3C1
SCHEMBL27687957 0.80 KCNH2 (1.00) KCNH2LMNASLC6A4HTR2B
Hydrochloric Acid SCHEMBL7701677 0.80 KCNH2 (0.57) KCNH2NR3C1
Hydrochloric Acid SCHEMBL27311830 0.79 KCNH2 (0.98) KCNH2SIGMAR1LMNASLC6A4HTR2B
SCHEMBL19668687 0.79 KCNH2 (0.55) KCNH2SCN4ASCN8ALMNACYP1A2
SCHEMBL12994787 0.79 KCNH2 (0.55) KCNH2SCN4ASCN8ALMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3494105-A2 COMPOUNDS AS INHIBITORS OF SODIUM CHANNELS Human Biomolecular Research Institute (US) 2019-06-12 EP disclosed
WO-2017210371-A2 COMPOUNDS AS INHIBITORS OF SODIUM CHANNELS HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2017-12-07 WO disclosed