SCHEMBL19669155

SCHEMBL19669155

CC(=O)[C@H]1[C@@H]2Cc3cc(OCc4cc(B5OC(C)(C)C(C)(C)O5)ccc4F)ccc3[C@@H]21

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.38
FFAR1 O14842 2/20 0.37
SCN3A Q9NY46 3/20 0.36
HIF1A Q16665 5/20 0.34
BACE1 P56817 1/20 0.33
BACE2 Q9Y5Z0 1/20 0.33
KCNH2 Q12809 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
MMP1 P03956 1/20 0.32
ADAM17 P78536 1/20 0.32
AAK1 Q2M2I8 1/20 0.31
MAOB P27338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18940276 0.93 FFAR1 (0.43) ROCK1FFAR1SCN3AHIF1ABACE1
SCHEMBL23927778 0.93 FFAR1 (0.43) ROCK1FFAR1SCN3AHIF1ABACE1
SCHEMBL18940306 0.93 FFAR1 (0.43) ROCK1FFAR1SCN3AHIF1ABACE1
SCHEMBL16845952 0.90 FFAR1 (0.38) ROCK1FFAR1SCN3AHIF1ABACE1
SCHEMBL29423910 0.90 FFAR1 (0.38) ROCK1FFAR1SCN3AHIF1ABACE1
SCHEMBL29423898 0.90 FFAR1 (0.38) ROCK1FFAR1SCN3AHIF1ABACE1
SCHEMBL15471420 0.87 FFAR1 (0.48) ROCK1FFAR1HIF1ABACE1BACE2
SCHEMBL18959381 0.81 FFAR1 (0.40) FFAR1SCN3AKCNH2MAOB
SCHEMBL23952751 0.79 SCN3A (0.39) ROCK1SCN3AHIF1ABACE1BACE2
SCHEMBL18940280 0.78 FFAR1 (0.44) FFAR1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9834563-B2 Antidiabetic substituted heteroaryl compounds MERCK SHARP & DOHME CORP. (US) 2017-12-05 US disclosed