SCHEMBL1967046

SCHEMBL1967046

CC(C)(CNC(=O)O)COc1cccc2ccc(-c3nnc4ccccn34)nc12

nearest known ligand 0.84

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 20/20 0.84
PIM2 Q9P1W9 20/20 0.84

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12589331 0.94 PIM1 (0.82) PIM1PIM2
SCHEMBL1976975 0.91 PIM1 (0.79) PIM1PIM2
SCHEMBL1967276 0.91 PIM1 (1.00) PIM1PIM2
SCHEMBL1965972 0.89 PIM1 (1.00) PIM1PIM2
Trifluoroacetic Acid SCHEMBL1976016 0.87 PIM1 (0.85) PIM1PIM2
SCHEMBL1966717 0.87 PIM1 (1.00) PIM1PIM2
SCHEMBL1980279 0.87 PIM1 (1.00) PIM1PIM2
SCHEMBL1976561 0.86 PIM1 (1.00) PIM1PIM2
SCHEMBL1966451 0.85 PIM1 (0.83) PIM1PIM2
SCHEMBL1975153 0.85 PIM1 (1.00) PIM1PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334677-A1 TRIAZOLOPYRIDINE COMPOUNDS AS PIM KINASE INHIBITORS Array Biopharma, Inc. (US) 2011-06-22 EP disclosed
WO-2010022076-A1 TRIAZOLOPYRIDINE COMPOUNDS AS PIM KINASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2010-02-25 WO disclosed