SCHEMBL19672731

SCHEMBL19672731

CSc1ccc(-c2cnc(N)c(-c3nnc(-c4ccccc4)o3)n2)cc1

nearest known ligand 0.79

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ATR Q13535 20/20 0.79
GSK3B P49841 1/20 0.65
PRKDC P78527 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13137928 0.89 ATR (1.00) ATRGSK3BPRKDC
SCHEMBL24248235 0.86 ATR (0.85) ATRGSK3BPRKDC
SCHEMBL2464265 0.84 ATR (0.85) ATRGSK3BPRKDC
SCHEMBL13137948 0.83 ATR (0.87) ATR
SCHEMBL2483805 0.82 ATR (1.00) ATR
SCHEMBL2512070 0.81 ATR (0.80) ATRGSK3BPRKDC
SCHEMBL2482305 0.81 ATR (1.00) ATRGSK3BPRKDC
SCHEMBL13138258 0.81 ATR (0.75) ATRGSK3BPRKDC
SCHEMBL2481994 0.81 ATR (1.00) ATR
SCHEMBL2504996 0.80 ATR (1.00) ATRGSK3BPRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4059932-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE Vertex Pharmaceuticals Incorporated (US) 2022-09-21 EP disclosed
EP-2376485-B1 PYRAZINE DERIVATIVES USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMA (US) 2017-12-06 EP disclosed